I-Retatrutide (LY3437943)iyi-peptide yokwenziwa yesizukulwane esilandelayo eyakhiwe njenge-i-agonist ye-receptor ephindwe kathathuihlose ama-receptor e-GLP-1, GIP, kanye ne-glucagon. Ukwakheka kwayo okusha kwama-molecule kuyayihlukanisa nobuchwepheshe be-peptide be-single- kanye ne-dual-receptor bangaphambilini, okwenza kube ngenye yamakhemikhali afundwe kabanzi ocwaningweni lwesimanje lwe-metabolic.
Inikezwa njengempuphu ehlanzekile kakhulu ene-lyophilized,I-Retatrutideinikeza ukuzinza okuhle kakhulu ekuphathweni kwelabhorethri, ukuthuthwa, kanye nokugcinwa kwesikhathi eside. Ivame ukusetshenziswa ocwaningweni lwesayensi oluhilela ukusabalalisa izimpawu ze-receptor, ukulawulwa kwe-metabolic, ubunjiniyela be-peptide, kanye nocwaningo lwe-endocrine.
✔ Ukuhlanzeka Okuphezulu (≥98% HPLC)
✔ I-Lyophilized Powder Emhlophe Kuya Kokumhlophe
✔ Ukuzinza Okuhle Kakhulu Kwezicelo Zocwaningo
✔ Ubuchwepheshe be-Agonist be-Triple Receptor
✔ Ukulawulwa Kwekhwalithi Okuqinile kanye Nokuhambisana Kweqembu
✔ Kufanelekela Ucwaningo Oluthuthukisiwe lwe-Peptide
| Into | Imininingwane |
|---|---|
| Igama Lomkhiqizo | I-Retatrutide |
| Igama elifanayo | LY3437943 |
| Ifomula Yamamolekyuli | C221H342N46O68* |
| Isisindo sama-molecule | Cishe 4731 Da* |
| Ukubukeka | I-White Lyophilized Powder |
| Ubumsulwa | ≥98% nge-HPLC |
| Isitoreji | Kunconywa -20°C |
| Ukuncibilika | Amanzi Ancibilikayo |
| Isicelo | Ucwaningo Lwelabhorethri Kuphela |
*Imininingwane ingahluka ngokuya ngeqoqo lokukhiqiza kanye nezindinganiso zokuhlaziya.
| Igama Lomkhiqizo | Inombolo ye-CAS |
|---|---|
| I-AOD-9604 | 221231-10-3 |
| I-BPC-157 | 137525-51-0 |
| I-PT-141 / i-Bremelanotide Acetate | 189691-06-3 |
| I-CJC-1295 | 863288-34-0 |
| I-GHK-Cu | 89030-95-5 |
| I-GHRP-2 | 158861-67-7 |
| I-Hexarelin | 140703-51-1 |
| IGF-1 LR3 | 946870-92-4 |
| I-Ipamorelin | 170851-70-4 |
| I-KPV / Alpha MSH (11-13) | 67727-97-3 |
| I-L-Arginine | 74-79-3 |
| I-MOTS-C | 1627580-64-6 |
| I-Oxytocin | 50-56-6 |
| I-PDA | 106-50-3 |
| I-Selank | 129954-34-3 |
| I-Semax | 80714-61-0 |
| I-Sermorelin | 86168-78-7 |
| I-SS-31 (Lyo) / I-Elamipretide | 736992-21-5 |
| Ingcezu ye-TB500 | 476014-70-7 |
| I-Tesamorelin | 218949-48-5 |
| I-Thymogen / i-Oglufanide | 38101-59-6 |
| I-Thymosin Alpha-1 / Thymalfasin | 62304-98-7 |
| I-Thymosin Beta-4 | 77591-33-4 |
| TB500 | 885340-08-9 |
| I-NVG-291 | 2135482-62-7 |
| I-CB4211 | 2361287-87-0 |
| I-DSIP | 62568-57-4 |
| I-Epitalon | 307297-39-8 |
| I-Gonadorelin | 33515-09-2 |
| LL-37 | 154947-19-0 |
| I-Melanotan II | 121062-08-6 |
| MK-0616 | 2249825-14-7 |
| I-NAD+ | 53-84-9 |
| I-Pamorelin | 57773-63-1 |
| I-PTD-DBM | 1241682-11-0 |
| Ingxenye 176-191 | 66004-57-7 |
| I-VIP | 40077-57-4 |
| I-PE-22-28 | 1136689-11-0 |
I-Retatrutide yenzelwe ukusebenza ngasikhathi sinye ama-receptor amathathu e-metabolic hormone:
Okuhlobene nokulawulwa kwesifiso sokudla, izindlela zokukhipha ukudla esiswini, kanye nezindlela zokuthumela izimpawu ezihlobene noshukela.
Kuhilelekile ekuzweleni izakhamzimba, ekudluliseni i-insulin, kanye nasezinqubweni zokulawula i-metabolic.
Kuhlobene nokusetshenziswa kwamandla, i-lipid metabolism, kanye nezindlela zokuzivumelanisa nezimo ze-metabolic.
Ukusebenza okuhlangene kwalezi zinhlelo ezintathu zama-receptor kwenza i-Retatrutide ibe yinkimbinkimbi yocwaningo yokuphenya ukusebenzisana okuyinkimbinkimbi kwe-metabolic kanye nezimpendulo zebhayoloji ezinemizila eminingi.
I-Retatrutide isibe yindaba ebalulekile ezindaweni eziningana zocwaningo lwesayensi, okuhlanganisa:
Abacwaningi bayaqhubeka nokuhlola iphrofayili yayo ehlukile ye-triple-agonist kanye nemiphumela engaba khona ekuthuthukisweni kwe-peptide yesikhathi esizayo.
Iqembu ngalinye le-Retatrutide kufanele lihlolwe ngokuhlaziya okujulile, okuhlanganisa:
Isitifiketi Sokuhlaziya (i-COA) singanikezwa uma siceliwe ukuqinisekisa ikhwalithi yomkhiqizo kanye nokulandeleka kwawo.
Ukuze kugcinwe ukuqina kwe-peptide okuhle kakhulu:
Isitoreji Sesikhathi Eside
Ngemva Kokwakhiwa Kabusha
Izimo zokugcina ezifanele zisiza ukugcina ubuqotho be-peptide kanye nokusebenza kokuhlaziya.
Izinketho zokupakisha ezitholakalayo zingafaka:
Ubuningi kanye nezinsizakalo zokupakisha ze-OEM ziyatholakala ezinhlanganweni zocwaningo ezifanelekayo.
I-Retatrutide inikezwa kuphela ngezinhloso zocwaningo lwelabhorethri kanye nokuhlaziya kuphela. Lo mkhiqizo awuvunyelwe ukusetshenziswa ngabantu, ukusetshenziswa kwezokwelapha, ukusetshenziswa kokwelapha, noma izinqubo zokuxilonga. Abacwaningi banesibopho sokuqinisekisa ukuhambisana nayo yonke imithethonqubo esebenzayo kanye neziqondiso zezikhungo.