149983567

I-Retatrutide (LY3437943) I-Peptide Powder – I-Peptide Yocwaningo Ehlanzekile Kakhulu

Incazelo emfushane:

✔ Ukuhlanzeka Okuphezulu ≥98% HPLC

✔ Ubuchwepheshe be-Agonist be-Triple Receptor

✔ Ukuzinza Okuhle Kakhulu Nokuncibilika

✔ Ukulawulwa Kwekhwalithi Okuqinile

✔ Ibanga Lokucwaninga Le-Lyophilized Powder

✔ Ukunikezwa Komhlaba Wonke Nokupakishwa Ngokwezifiso


Imininingwane Yomkhiqizo

Amathegi Omkhiqizo

Ukubuka Konke Komkhiqizo

I-Retatrutide (LY3437943)iyi-peptide yokwenziwa yesizukulwane esilandelayo eyakhiwe njenge-i-agonist ye-receptor ephindwe kathathuihlose ama-receptor e-GLP-1, GIP, kanye ne-glucagon. Ukwakheka kwayo okusha kwama-molecule kuyayihlukanisa nobuchwepheshe be-peptide be-single- kanye ne-dual-receptor bangaphambilini, okwenza kube ngenye yamakhemikhali afundwe kabanzi ocwaningweni lwesimanje lwe-metabolic.

Inikezwa njengempuphu ehlanzekile kakhulu ene-lyophilized,I-Retatrutideinikeza ukuzinza okuhle kakhulu ekuphathweni kwelabhorethri, ukuthuthwa, kanye nokugcinwa kwesikhathi eside. Ivame ukusetshenziswa ocwaningweni lwesayensi oluhilela ukusabalalisa izimpawu ze-receptor, ukulawulwa kwe-metabolic, ubunjiniyela be-peptide, kanye nocwaningo lwe-endocrine.


Izici Eziyinhloko

✔ Ukuhlanzeka Okuphezulu (≥98% HPLC)

✔ I-Lyophilized Powder Emhlophe Kuya Kokumhlophe

✔ Ukuzinza Okuhle Kakhulu Kwezicelo Zocwaningo

✔ Ubuchwepheshe be-Agonist be-Triple Receptor

✔ Ukulawulwa Kwekhwalithi Okuqinile kanye Nokuhambisana Kweqembu

✔ Kufanelekela Ucwaningo Oluthuthukisiwe lwe-Peptide


Imininingwane Yomkhiqizo

Into Imininingwane
Igama Lomkhiqizo I-Retatrutide
Igama elifanayo LY3437943
Ifomula Yamamolekyuli C221H342N46O68*
Isisindo sama-molecule Cishe 4731 Da*
Ukubukeka I-White Lyophilized Powder
Ubumsulwa ≥98% nge-HPLC
Isitoreji Kunconywa -20°C
Ukuncibilika Amanzi Ancibilikayo
Isicelo Ucwaningo Lwelabhorethri Kuphela

*Imininingwane ingahluka ngokuya ngeqoqo lokukhiqiza kanye nezindinganiso zokuhlaziya.

Igama Lomkhiqizo Inombolo ye-CAS
I-AOD-9604 221231-10-3
I-BPC-157 137525-51-0
I-PT-141 / i-Bremelanotide Acetate 189691-06-3
I-CJC-1295 863288-34-0
I-GHK-Cu 89030-95-5
I-GHRP-2 158861-67-7
I-Hexarelin 140703-51-1
IGF-1 LR3 946870-92-4
I-Ipamorelin 170851-70-4
I-KPV / Alpha MSH (11-13) 67727-97-3
I-L-Arginine 74-79-3
I-MOTS-C 1627580-64-6
I-Oxytocin 50-56-6
I-PDA 106-50-3
I-Selank 129954-34-3
I-Semax 80714-61-0
I-Sermorelin 86168-78-7
I-SS-31 (Lyo) / I-Elamipretide 736992-21-5
Ingcezu ye-TB500 476014-70-7
I-Tesamorelin 218949-48-5
I-Thymogen / i-Oglufanide 38101-59-6
I-Thymosin Alpha-1 / Thymalfasin 62304-98-7
I-Thymosin Beta-4 77591-33-4
TB500 885340-08-9
I-NVG-291 2135482-62-7
I-CB4211 2361287-87-0
I-DSIP 62568-57-4
I-Epitalon 307297-39-8
I-Gonadorelin 33515-09-2
LL-37 154947-19-0
I-Melanotan II 121062-08-6
MK-0616 2249825-14-7
I-NAD+ 53-84-9
I-Pamorelin 57773-63-1
I-PTD-DBM 1241682-11-0
Ingxenye 176-191 66004-57-7
I-VIP 40077-57-4
I-PE-22-28 1136689-11-0

Indlela Yokusebenza

I-Retatrutide yenzelwe ukusebenza ngasikhathi sinye ama-receptor amathathu e-metabolic hormone:

Isamukeli se-GLP-1

Okuhlobene nokulawulwa kwesifiso sokudla, izindlela zokukhipha ukudla esiswini, kanye nezindlela zokuthumela izimpawu ezihlobene noshukela.

Isamukeli se-GIP

Kuhilelekile ekuzweleni izakhamzimba, ekudluliseni i-insulin, kanye nasezinqubweni zokulawula i-metabolic.

I-Glucagon Receptor

Kuhlobene nokusetshenziswa kwamandla, i-lipid metabolism, kanye nezindlela zokuzivumelanisa nezimo ze-metabolic.

Ukusebenza okuhlangene kwalezi zinhlelo ezintathu zama-receptor kwenza i-Retatrutide ibe yinkimbinkimbi yocwaningo yokuphenya ukusebenzisana okuyinkimbinkimbi kwe-metabolic kanye nezimpendulo zebhayoloji ezinemizila eminingi.


Izicelo Zocwaningo

I-Retatrutide isibe yindaba ebalulekile ezindaweni eziningana zocwaningo lwesayensi, okuhlanganisa:

  • Izifundo zendlela ye-Metabolic
  • Ucwaningo lokubonisana kwama-receptor e-Peptide
  • Uphenyo lwesistimu ye-endocrine
  • Ucwaningo lwe-homeostasis yamandla
  • Amamodeli ocwaningo lokukhuluphala kanye nokuphazamiseka kwe-metabolic
  • Izifundo zobudlelwano besakhiwo nomsebenzi
  • Amaphrojekthi obunjiniyela be-peptide athuthukisiwe

Abacwaningi bayaqhubeka nokuhlola iphrofayili yayo ehlukile ye-triple-agonist kanye nemiphumela engaba khona ekuthuthukisweni kwe-peptide yesikhathi esizayo.


Ukuqinisekisa ikhwalithi

Iqembu ngalinye le-Retatrutide kufanele lihlolwe ngokuhlaziya okujulile, okuhlanganisa:

  • I-Chromatography Yoketshezi Esebenza Kakhulu (i-HPLC)
  • I-Mass Spectrometry (MS)
  • Ukuqinisekiswa Kokubukeka
  • Ukuhlolwa Kobumsulwa
  • Ukuhlolwa Kokuhambisana Kweqembu

Isitifiketi Sokuhlaziya (i-COA) singanikezwa uma siceliwe ukuqinisekisa ikhwalithi yomkhiqizo kanye nokulandeleka kwawo.


Isitoreji Nokuphathwa

Ukuze kugcinwe ukuqina kwe-peptide okuhle kakhulu:

Isitoreji Sesikhathi Eside

  • Gcina ku--20°C noma ngaphansi
  • Vikela ekukhanyeni okuqondile
  • Gcina isitsha sivalwe kahle

Ngemva Kokwakhiwa Kabusha

  • Landela izinqubo zokuphatha ilabhorethri
  • Nciphisa imijikelezo yokuqandisa nokuncibilikisa ephindaphindwayo
  • Sebenzisa izihlanzi ezifanele zokuhlola ezihlanzekile

Izimo zokugcina ezifanele zisiza ukugcina ubuqotho be-peptide kanye nokusebenza kokuhlaziya.


Izinketho Zokupakisha

Izinketho zokupakisha ezitholakalayo zingafaka:

  • 2mg/iVili
  • 5mg/iVili
  • 10mg/iVili
  • 15mg/iVili
  • Ukupakishwa Ngokwezifiso Kuyatholakala

Ubuningi kanye nezinsizakalo zokupakisha ze-OEM ziyatholakala ezinhlanganweni zocwaningo ezifanelekayo.


Isihlangululo

I-Retatrutide inikezwa kuphela ngezinhloso zocwaningo lwelabhorethri kanye nokuhlaziya kuphela. Lo mkhiqizo awuvunyelwe ukusetshenziswa ngabantu, ukusetshenziswa kwezokwelapha, ukusetshenziswa kokwelapha, noma izinqubo zokuxilonga. Abacwaningi banesibopho sokuqinisekisa ukuhambisana nayo yonke imithethonqubo esebenzayo kanye neziqondiso zezikhungo.


  • Okwedlule:
  • Olandelayo:

  • Bhala umlayezo wakho lapha bese uwuthumela kithi